AnnoTitoloTipo MIUR
2025Modelling-filtered drug repurposing and first-in-protein SPR validation of histone deacetylase 4 inhibitors for Ataxia-telangiectasia
(BIOMÉDECINE & PHARMACOTHÉRAPIE)
Articolo in rivista
2024Recent Applications of In Silico Approaches for Studying Receptor Mutations Associated with Human Pathologies
(MOLECULES)
Articolo in rivista
2023Identification of a novel adiponectin receptor and opioid receptor dual acting agonist as a potential treatment for diabetic neuropathy
(BIOMÉDECINE & PHARMACOTHÉRAPIE)
Articolo in rivista
2021Peptidomimetics in Silico
(MOLECULAR INFORMATICS)
Articolo in rivista
2020In-silico design and biological investigations of Diabetic Neuropathy modulators: could MOR become a focal mediator for this pathology?Contributo in Atti di convegno
2020Interaction of natural flavonoid eriocitrin with beta-cyclodextrin and hydroxypropyl-beta-cyclodextrin: an NMR and molecular dynamics investigation
(NEW JOURNAL OF CHEMISTRY)
Articolo in rivista
2020Parameters for irreversible inactivation of monoamine oxidase
(MOLECULES)
Articolo in rivista
2020Pharmacological properties and biochemical mechanisms of MOR ligands might be due to different binding poses. MD Studies
(FUTURE MEDICINAL CHEMISTRY)
Articolo in rivista
2020Quantum chemical and molecular dynamics studies of MUC-1 calix[4,8]arene scaffold based anti-cancer vaccine candidates
(JOURNAL OF CHEMICAL INFORMATION AND MODELING)
Articolo in rivista
2019Exploring the biological activity of a library of 1,2,5-oxadiazole derivatives endowed with antiproliferative activity
(ANTICANCER RESEARCH)
Articolo in rivista
2019Molecular modeling and biological studies show that some μ-opioid receptor agonists might elicit analgesia acting as MMP-9 inhibitors
(FUTURE MEDICINAL CHEMISTRY)
Articolo in rivista
2018In silico screening for human norovirus antivirals reveals a novel non-nucleoside inhibitor of the viral polymerase
(SCIENTIFIC REPORTS)
Articolo in rivista
2018ML10302Monografia o trattato scientifico
2018Molecular modeling studies on mu opioid receptor of agonists and antagonists, endogenous and exogenous, ligandsPoster
2017A field-based disparity analysis of new 1,2,5- oxadiazole derivatives endowed with antiproliferative activity
(CHEMICAL BIOLOGY & DRUG DESIGN)
Articolo in rivista
2017Correlating in Vitro Target-Oriented Screening and Docking: Inhibition of Matrix Metalloproteinases Activities by Flavonoids
(PLANTA MEDICA)
Articolo in rivista
2017Design, synthesis and docking study of novel coumarin ligands as potential selective acetylcholinesterase inhibitors
(JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY)
Articolo in rivista
2017Homology-based modeling of rhodopsin-like family members in the inactive state: structural analysis and deduction of tips for modeling and optimization.
(MOLECULAR INFORMATICS)
Articolo in rivista
2016How to choose the suitable template for homology modelling of GPCRs: 5-HT7 receptor as a test case
(MOLECULAR INFORMATICS)
Articolo in rivista
2016Rescuing Abandoned Molecules as Nav1.7 and PCSK9 Inhibitors
(JOURNAL OF ADVANCES IN MEDICAL AND PHARMACEUTICAL SCIENCES)
Articolo in rivista
2016Tips for modelling histamine receptors
(INFLAMMATION RESEARCH)
Abstract in Atti di convegno
2015How does binding of imidazole-based inhibitors to heme oxygenase-1 influence their conformation? Insights combining crystal structures and molecular modelling
(ACTA CRYSTALLOGRAPHICA. SECTION B, STRUCTURAL SCIENCE, CRYSTAL ENGINEERING AND MATERIALS)
Articolo in rivista
2015Identification of essential residues for binding and activation in the human 5-HT7(a) serotonin receptor by molecular modeling and site-directed mutagenesis
(FRONTIERS IN BEHAVIORAL NEUROSCIENCE)
Articolo in rivista
2015Identification of 5-Methoxyflavone as a Novel DNA Polymerase-Beta Inhibitor and Neuroprotective Agent against Beta-Amyloid Toxicity.
(JOURNAL OF NATURAL PRODUCTS)
Articolo in rivista
2015In silico identification and pharmacological evaluation of 5-methoxyflavone as a neuroprotective agent against β-amyloid-induced toxicityAbstract in Atti di convegno
2015Neuroprotective effects of the monoamine oxidase inhibitor tranylcypromine and its amide derivatives against Aβ(1-42)-induced toxicity
(EUROPEAN JOURNAL OF PHARMACOLOGY)
Articolo in rivista
2015Potential of Aryl-urea-Benzofuranylthiazoles hybrids as multitasking agents in Alzheimer’s disease
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
20155HT1a Receptor Binding Affinities of a Series of Serotonin Transporter (SERT) Inhibitors and Related Thermodynamic Insights
(JOURNAL OF ADVANCES IN MEDICAL AND PHARMACEUTICAL SCIENCES)
Articolo in rivista
2014Computational Comparison of Imidazoline Association with the I2 Binding Site in Human Monoamine Oxidases
(JOURNAL OF CHEMICAL INFORMATION AND MODELING)
Articolo in rivista
2014Correction to Computational Comparison of imidazoline association with the i2 binding site in human monoamine oxidases (Journal of Chemical Information and Modeling (2014) 54:4 (1200-1207))
(JOURNAL OF CHEMICAL INFORMATION AND MODELING)
Articolo in rivista
2014Sequential application of ligand and structure based modeling approaches to index chemicals for their hH4R antagonism
(PLOS ONE)
Articolo in rivista
2013Heme Oxygenase 1 and Heme Oxygenase 2 as druggable targets: doching and two hybrid system to identifying and characterizing protein-protein interactionsAbstract in Atti di convegno
2013Heme Oxygenase 1 and Heme Oxygenase 2 As Druggable Targets: Docking and Two Hybrid System To Identifying and Characterizing Protein-Proten Interactions.Contributo in Atti di convegno
2013Heme oxygenase-1 and Heme oxygenase-2 as druggable targets: Docking and two-hybrid system to identify and characterize protein-protein interactionPoster
2013Heme oxygenase-2/adiponectin protein-protein interaction in metabolic syndrome
(BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS)
Articolo in rivista
2013Stereoretentive Chlorination of Cyclic Alcohols Catalyzed by Titanium (IV) Tetrachloride: Evidence for a Front Side Attack Mechanism.
(JOURNAL OF ORGANIC CHEMISTRY)
Articolo in rivista
2012Evaluation of Imidazole-Based Compounds as Heme Oxygenase-1 Inhibitors
(CHEMICAL BIOLOGY & DRUG DESIGN)
Articolo in rivista
2012Imidazole Derivatives as Heme Oxygenase-1 InhibitorsPoster
2012Imidazole Derivatives as Heme Oxygenase-1 InhibitorsAbstract in Atti di convegno
2012Imidazole Derivatives as Heme Oxygenase-1 InhibitorsContributo in Atti di convegno
2012Molecular modelling and site-directed mutagenesis reveal essential residues for 5-HT7 receptor bindingAbstract in Atti di convegno
2012Sulfonilamidothiopyrimidone and thiopyrimidone derivatives as selective COX-2 inhibitors: Synthesis, biological evaluation, and docking studies
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2012Synthesis, benzodiazepine receptor binding and molecular modelling of isochromeno[4,3-c]pyrazol-5(1H)-one derivatives
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2011Drug delivery of synthetic antisense “Bioconjugates” for anticancer therapy DNA.
(EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES)
Contributo in Atti di convegno
2011DRUG DELIVERY OF SYNTHETIC ANTISENSE-DNA "BIOCONJUGATES" FOR ANTICANCER THERAPY
(EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES)
Articolo in rivista
2011Drug Delivery of Synthetic Antisense-DNA “bioconjugates” for Anticancer Therapy
(EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES)
Poster
2011Novel Benzo[b]thiophene Derivatives as New Potential Antidepressants with Rapid Onset of Action
(JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2011Spectroscopic Investigation and Molecular Modeling on Porphyrin/PAMAM Supramolecular Adduct
(PHOTOCHEMISTRY AND PHOTOBIOLOGY)
Articolo in rivista
2010Potential immunoregulatory role of heme oxygenase-1 in human milk: a combined biochemical and molecular modeling approach
(JOURNAL OF NUTRITIONAL BIOCHEMISTRY)
Articolo in rivista
2009Potential of the nature's biochemistry for for drug designContributo in Atti di convegno
2009TCP-FA4: A derivative of tranylcypromine showing improved blood-brain permeability
(BIOCHEMICAL PHARMACOLOGY)
Articolo in rivista
2008Computational studies on the role of human milk heme oxygenase as immuno modulating factorContributo in Atti di convegno
2008Identification of novel scaffolds leading to small molecole DNA polymerase-β inhibitors with potential in neurodegenerative and oncology disordersContributo in Atti di convegno
2008Sensory Analysis on Red Wines: Discrimination by Adaptive Fuzzy Partition (AFP)
(JOURNAL OF SENSORY STUDIES)
Articolo in rivista
2008The cell cycle molecules behind neurodegeneration in Alzheimer's disease: perspectives for drug development
(CURRENT MEDICINAL CHEMISTRY)
Articolo in rivista
2008The shape of the flavin in monoamine oxidaseContributo in Atti di convegno
2008Theoretical calculations of the catalytic triad in short chain alcohol dehydrogenases/reductases
(BIOPHYSICAL JOURNAL)
Articolo in rivista
200816. Towards a complete picture of chiral discrimination processes by C9 carbamate derivatives of dihydroquinine: interaction mechanisms of diastereoisomeric 9-O-[(S)- or (R)-1-(1-naphthyl)ethylcarbamate]dihydroquinine and the two enantiomers of N-(3,5-dinitrobenzoyl)alanine methyl ester
(TETRAHEDRON-ASYMMETRY)
Articolo in rivista
2007Docking simulation of complex between 2,5-xilidine and Rigidoporus lignosus laccaseContributo in Atti di convegno
2007DUAL 5-HT1A or 5-HT7 RECEPTOR LIGANDS-SERT BLOCKERS. IMPLICATIONS FOR LIGAND-SELECTIVE RECEPTOR CONFORMATIONS: PHENOTYPE BASED SELECTIVITYContributo in Atti di convegno
2007Interactions of imidazoline ligands with the active site of purified monoamine oxidase A
(THE FEBS JOURNAL)
Articolo in rivista
2007Models of imidazoline isomers in the active site of monoamine oxidase BContributo in Atti di convegno
2007Molecular modelling of a novel class of N5-methanesulfonamide dihydrothienopyrimidinoners as potential dual COX-2 inhibitor/Contributo in Atti di convegno
2007NEW APPROACHES TO ANTICANCER THERAPYContributo in Atti di convegno
2006Binding of imidazline ligands to the active site of purified MAO AContributo in Atti di convegno
2006Comparing Log P Calculations by the Ghose-Crippen and Villar MethodsContributo in volume (Capitolo o Saggio)
2006DESIGN AND SYNTHESIS OF MULTIPLE LIGANS: NEW ARYLAMINES AND THEIR BINDING AFFINITY TOWARD 5-HT TRANSPORTER (SERT) AND 5-HT7- RECEPTORSContributo in Atti di convegno
2006Editorial: Usefulness and robustness of In Silico and experimental technology for drug discovery
(CURRENT PHARMACEUTICAL DESIGN)
Articolo in rivista
2006Emerging antifungal azoles and effects on Magnaporthe grisea
(MYCOLOGICAL RESEARCH)
Articolo in rivista
2006Enhancement of drug affinity for cell membranes by conjugation with lipoamino acids II. Experimental and computational evidence using biomembrane models
(INTERNATIONAL JOURNAL OF PHARMACEUTICS)
Articolo in rivista
2006GraphBlast: A Fast and Universal Method for Querying GraphsContributo in Atti di convegno
2006Molecular modelling of a novel class of N5-methanesulfonamide dihydrothienopyrimidinoners as as potential dual COX-2 inhibitor/nitric oxide anti-releasing agents
(MEDICINAL CHEMISTRY RESEARCH)
Articolo in rivista
2006Structural data: the basis for molecular modellingContributo in volume (Capitolo o Saggio)
2006Substrate and inhibitor specificity of class 1 and class 2 histone deacetylases
(JOURNAL OF BIOTECHNOLOGY)
Articolo in rivista
2005Combined NMR-crystallographic and modelling investigation of the inclusion of molsidomine into alpha-, beta - and gamma -cyclodextrins
(BIOORGANIC & MEDICINAL CHEMISTRY)
Articolo in rivista
2005Enhancement of drug affinity for cell membranes by conjugation with lipoamino acids. I. Synthesis and biological evaluation of lipophilic conjugates of tranylcypromine
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2005Hydrophobic molecular similarity from MST fractional contributions to the octanol/water partition coefficient
(JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN)
Articolo in rivista
2005Molecular properties of ibuprofen and its solid dispersion with Eudragit RL100 studied by solid-state Nuclear Magnetic Resonance
(PHARMACEUTICAL RESEARCH)
Articolo in rivista
2005Pyrazole Derivatives as Photosynthetic Electron TransportInhibitors: New Leads and Structure Activity Relationship
(JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY)
Articolo in rivista
2005The Catalyric Mechanism of Short-Chain Dehydrogenase/ReductasesContributo in Atti di convegno
2004COMBINING NMR AND MOLECULAR MODELLING IN A DRUG DELIVERY CONTEXT: investigation of the multi-mode inclusion of a new NPY-5 antagonist bromobenzenesulfonamide into beta-cyclodextrin
(BIOORGANIC & MEDICINAL CHEMISTRY)
Articolo in rivista
2004Lipophilic conjugates of methotrexate with short-chain alkylamino acids as DHFR inhibitors. Synthesis, biological evaluation, and molecular modeling
(BIOORGANIC & MEDICINAL CHEMISTRY)
Articolo in rivista
2004Lipophilic conjugates of methotrexate with short-chain alkylaminoacids as DHFR inhibithors. Synthesis, biological avaluation, and molecular modeling
(BIOORGANIC & MEDICINAL CHEMISTRY)
Articolo in rivista
2004Molecular Modelling of endothelin ETA and ETBContributo in Atti di convegno
2004Solid state NMR of drugs: A Study of Non-steroidal Anti-infammatory drugs and Their dispersions with polymer carriersContributo in Atti di convegno
2004Solid state NMRof drugs: a study of non-steroidal anti-inflammatory drugs and their dispersions with polymeric carriersContributo in Atti di convegno
2004Study of structural and dynamic behaviour of ibuprofen and its solid dispersions with eudragit RL100 by means of solid state NMRContributo in Atti di convegno
20045-HT1A receptor binding analysis of thienopyrimidinones partial agonists: a paradigm breaking study regarding the pharmacophoric leadership of the protonated piperazine ring in GPCR ligandsAbstract in Atti di convegno
2003Carbohydrate-Ligand Complex Binding: EMPIRICAL FREE ENERGY MODELINGContributo in Atti di convegno
2003Determination of orientation of DNA-antimetabolites in the real receptor cavity using 3D QSAR method BiSContributo in Atti di convegno
2003Hydrophobic Similarity between Molecules: A MST-Based Hydrophobic Similarity Index and its application to Drug Design and Drug Delivery StudiesContributo in Atti di convegno
2003Parallel version of MultiGenContributo in Atti di convegno
2003Study of structural and dynamic behaviour of ibuprofen and its complexes with Eudragit® RL100 by means of solid state NMRContributo in Atti di convegno
2003STUDY OF STRUCTURAL AND DYNAMIC BEHAVIOUR OF IBUPROFEN AND ITS COMPLEXES WITH EUDRAGIT® RL100 BY NERANS OF SOLID STATEContributo in Atti di convegno
2003WINDOWS TO THE WORLD OF LIGANDS-MACROMOLECULAR RECEPTOR INTERACTIONSContributo in Atti di convegno
2002Combining molecular modeling with experimental methodologies: mechanism of membrane permeation and accumulation of ofloxacin
(BIOORGANIC & MEDICINAL CHEMISTRY)
Articolo in rivista
2002COMPARING A BIS (BIOLOGICAL SUBSTRATE SEARCH) ALIGNMENT OF ANTICANCER DNA AND DNA/RNA ANTIMETABOLITES INTO THEIR ACTIVE SITES WITH .PDB CO-CRYSTALSContributo in Atti di convegno
2002Crystallographic, NMR and ab initio calculation studies of tautomerism among substituted dihydrothiazol-2-ylhydrazones
(JOURNAL OF THE CHEMICAL SOCIETY. PERKIN TRANSACTIONS 2)
Articolo in rivista
2002Crystallographic, NMR and ab initio calculation studies of tautomerism among substituted thiazol-2-yl-hydrazines
(JOURNAL OF THE CHEMICAL SOCIETY. PERKIN TRANSACTIONS 2)
Articolo in rivista
2002Molecular modelling of lipophilic conjugates of methotrexate with lipoamino acidsContributo in Atti di convegno
2002MOLECULAR MODELLING OF LIPOPHILIC CONJUGATES OF METHOTREXATE WITH LIPOAMONI ACIDSContributo in Atti di convegno
2002Molecular Modelling of non-steroidal antiinflammatory drugs in Eudragit Retard polymers solid dispersionsContributo in Atti di convegno
2002Multi-conformational method of analysis of biological activity of molecular structures
(JOURNAL OF STRUCTURAL CHEMISTRY)
Articolo in rivista
2002Synthesis and molecular modelling of new 1-(aryl)-3-4-(aryl)piperazin-1-yl-1-propane derivatives with high affinity at the serotonin transporter and at 5-HT1A receptors
(JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2002Whoever sits at the bottom of a well to contemplate the sky, will find it small
(CURRENT PHARMACEUTICAL DESIGN)
Articolo in rivista
20024 Methyl-2-[N-(3,4-methylenedioxy-benzylidene)hydrazino]thiazole and its reduction product, 4-methyl-2-[N-(3,4-methylenedioxybenzylidene)-hydrazono]-4,5-dihydrothiazole
(ACTA CRYSTALLOGRAPHICA. SECTION C, CRYSTAL STRUCTURE COMMUNICATIONS)
Articolo in rivista
2001A method for determination of form and sizes of pocket in "receptor-ligand" complexesContributo in Atti di convegno
2001A 3D QSAR study of Monoamino Oxidase B inhibitors, using the chemical function based pharmacophore generation approach
(JOURNAL OF ENZYME INHIBITION)
Articolo in rivista
2001An Alternative Method for 3D-QSAR and the Alignment of Molecular Structures: BiS (Biological Substrate Search)Contributo in Atti di convegno
2001Current pharmaceutical design: Preface
(CURRENT PHARMACEUTICAL DESIGN)
Articolo in rivista
2001Design, synthesis and binding properties of novel and selective 5-HT3 and 5-HT4 receptor ligands
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2001From Molecular Spectra to Biological Activities: a Comparative Spectra Analysis (CoSA) study on Epidermal Growth Factor Receptor Protein Tyrosine Kinase InhibitorsContributo in Atti di convegno
2001MULTIGEN: A NEW PARADIGM FOR “MULTICONFORMATIONAL” ALIGNMENT OF MOLECULAR STRUCTURES IN 3D-QSAR STUDIESContributo in Atti di convegno
2001New 3D-QSAR Algorithm BiS for orientation and alignment of molecules to receptor. Analysis of anti-tubercular action of podandsContributo in Atti di convegno
2001Potential of Pyrazolooxadiazinone Derivatives as Serine Protease Inhibitors
(JOURNAL OF ENZYME INHIBITION)
Articolo in rivista
2001Preparation, characterisation and photosensitivity studies of solid dispersions of diflunisal and Eudragit RS100 (R) and RL100 (R)
(INTERNATIONAL JOURNAL OF PHARMACEUTICS)
Articolo in rivista
2000CoMFA study of new acetyl-coa: cholesterol o-acyl transferase (ACAT) inhibitors
(SCIENTIA PHARMACEUTICA)
Articolo in rivista
2000Conformational analysis and pharmacophore identification of new serotonin 5-HT4 receptor ligands made by DISCOAbstract in Atti di convegno
2000PARM mapping of rat and human serotonin 1A (5-HT1A) receptorAbstract in Atti di convegno
20003D-QSAR study of new acetyl-COA:cholesterol O-acyl transferase (ACAT) inhibitors
(SCIENTIA PHARMACEUTICA)
Articolo in rivista
20003D-QSAR Using ”Multiconformer” Alignment: The Use of HASL in the Analysis of 5-HT1A Thienopyrimidinone Ligands
(JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN)
Articolo in rivista
1999Combining different 3D-QSAR methodologies in a multiconformer context: a new approach to map not X-ray determined targets of pharmaceutical interest overcoming alignment problemsContributo in Atti di convegno
1999Receptor modeling using " Multiconformer" alignment: comparison of HASL and CoMFA in the analysis of 5-HT1A thienopyrimidinone ligandsAbstract in Atti di convegno
1999Thiazole derivatives as inhibitors of purified bovine liver mitochondrial monoamine oxidase-B: structure-activity relationships and theoretical study
(JOURNAL OF ENZYME INHIBITION)
Articolo in rivista
1998Application of PARM to constructing and comparing 5-HT1A and alfa1 receptor modelsContributo in Atti di convegno
1998Application of Parm to constructing and comparing 5-HT1A and alfa1 receptor modelsAbstract in Atti di convegno
1998Application of PARM to constructing and comparing 5-HT1A and alpha1 receptor modelsContributo in Atti di convegno
1998Building a model of interaction at the NK-2 receptors: Polycondensed heterocycles containing the pyrimidoindole skeleton
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
1998Building a model of interaction at the NK-2 receptors: polycondensed heterocycles containing the pyrimidoindole skeleton
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
1998De Novo Design of Inhibitors of Protein Tyrosine Kinase pp60c-srcContributo in Atti di convegno
1998Determination of the cholecalciferol-lipid complex using a combination of comparative modelling and nmr spectroscopyContributo in Atti di convegno
19985-HT1A receptors mapping by conformational analysis (2D NOESY/MM) and ”three way modelling” (HASL, CoMFA, PARM)Contributo in Atti di convegno
19985-HT1A receptors mapping by conformational analysis (2D NOESY/MM) and "tree way modelling" (HASL, CoMFA, PARM)Abstract in Atti di convegno
1997Study on new neurokinin antagonists: polycondensed heterocycles containing the indole skeleton
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
1997Synthesis and pharmacological evaluation of benzothieno and [1]pyridothieno [2,3-d]triazole derivatives as antagonists at NK-1 receptorsContributo in Atti di convegno
1997Synthesis of 1-phenyl-6-arilsubstituted pyrazolopyrimidothiazole as antagonists at the NK-2 receptorsAbstract in Atti di convegno
1996Alkylation of non-electron rich nitrogen heterocycles by alkyl orthoformates: quantum chemistry calculations
(JOURNAL OF HETEROCYCLIC CHEMISTRY)
Articolo in rivista
1996Identification of an impurity in the synthesis of pharmacologically active pyrazolotriazolopyrimidines by a combined spectrometric approach
(RAPID COMMUNICATIONS IN MASS SPECTROMETRY)
Articolo in rivista
1996Synthesis and COMFA study of new heterocyclic compounds as potential AcylCoA: cholesterol O-acyltransferase inhibitorsContributo in Atti di convegno
1996Synthesis and NK-2 antagonist effect of 1,6-diphenyl-pyrazolo [3, 4-d]-thiazolo[3,2-a]4H-pyrimidin-4-one
(BIOORGANIC & MEDICINAL CHEMISTRY LETTERS)
Articolo in rivista
1996Synthesis of 3-methyl substituted pyrazolotriazolopyrimidin-4-one and pyrazolo-thiazolopyrimidin-4-one derivatives
(JOURNAL OF HETEROCYCLIC CHEMISTRY)
Articolo in rivista
1995CoMFA contributions to a binding mode for NK2 receptor antagonistsAbstract in Atti di convegno
1995Heterocyclic systems containing the pyrimido-2,4-dione ring as selective ligands for the alpha1-adrenoceptorsContributo in Atti di convegno
1995Potential of alkyl orthoformates as alkylating agents of non-electron rich nitrogen heterocycles
(JOURNAL OF HETEROCYCLIC CHEMISTRY)
Articolo in rivista
1995Potential of indole skeleton containing heterocycles as antagonists at the neurokinin (NK) receptor systemAbstract in Atti di convegno
1995Unforeseen alkylating effect of triethylorthoformate in the synthesis of pyrazolotriazolopyrimidine derivatives
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
1994A new procedure for the synthesis of 4H-pyrazolo[1,5-c][1,3,5]thiadiazine-4-thiones
(JOURNAL OF HETEROCYCLIC CHEMISTRY)
Articolo in rivista
1994Study on the tachykinins antagonist effect of combinatorial functionalized heterocycle replacements in tryciclic pyrimidine derivativesAbstract in Atti di convegno
1994Synthesis of new thiazinoindole derivatives and their evaluation as inhibitors of human leukocyte elastase and other related serine proteases
(BIOORGANIC & MEDICINAL CHEMISTRY LETTERS)
Articolo in rivista
1993An efficient procedure for the synthesis of Pyrazolo[3,4-d] [1,3] Thiazin-4-ones
(HETEROCYCLES)
Articolo in rivista
1993Pyrazolothiazolopyrimidine derivatives as novel class of anti-inflammatory or antinociceptive agents: synthesis, structural characterization and pharmacological evaluation
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
1993Pyrazolothiazolopyrimidine derivatives as a novel class of anti-inflammatory or antinociceptive agents: synthesis, structural characterization and pharmacological evaluation
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
1993Pyrimido [5,4-b] benzofuran and pyrimido [5,4-b] benzothiophene derivatives. Ligands for alpha1- and 5HT1A- receptors
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
1992Synthesis and pharmacological properties of pyrazolotriazolopyrimidine derivatives
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
1991Pyrimido[5,4-b] Indole derivatives. 1. A new class of potent and selective alpha-1 adrenoceptor ligands
(JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
1991Synthesis and pharmacological evaluation of pyrazolopyrimidobenzoxazole and pyrazolopyrimidobenzothiazole derivatives
(BOLLETTINO CHIMICO FARMACEUTICO)
Articolo in rivista
1990Synthesis and pharmacological activity of 6H-thiazolo[3’,2’:1,2]-5-oxopyrimido[5,4-b] Indole derivatives, a new heterocyclic ring system
(PHARMAZIE)
Articolo in rivista
1988New heterocyclic ring systems. Synthesis and pharmacological activity of 6H-1,3,4-thiadiazolo [3’,2’: 1,2]-5-oxopyrimido[5,4-b]indole derivatives and of 1-phenyl-6H-1,2,4-Triazolo [1’,5’: 1,2]-5-oxopyrimido [5,4-b]Indole
(IL FARMACO. EDIZIONE SCIENTIFICA)
Articolo in rivista
IN STAMPATherapeutically valuable bioactive extracts from Mediterranean plants: green technologies and molecolar modelling for viable endeavour.Contributo in volume (Capitolo o Saggio)